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API原料药

Intermediates中间体

杂质列表

API原料药

API 原料药

No.

Product Name

中文品名

Specification

CAS No.

1.

Asenapine Maleate

阿森那平马来酸盐

99%

85650-56-2

2.

Apremilast

阿普斯特

99%

608141-41-9

3.

Acotiamide hydrochloride trihydrate

盐酸阿考替胺三水合物

99%

773092-05-0

4.

Aripiprazole lauroxil

月桂酰阿立哌唑

99%

1259305-29-7

5.

Alvimopan

爱维莫潘

99%

156053-89-3

6.

Bepotastine besylate

苯磺酸贝托司汀

99%

190786-44-8

7.

Dronedarone hydrochloride

盐酸决奈达隆

99%

141625-93-6

8.

Deferasirox

地拉罗司

99%

201530-41-8

9.

Dabigatran etexilate mesylate

达比加群酯甲磺酸盐

99%

872728-81-9

10.

Edoxaban tosylate monohydrate

依度沙班对甲苯磺酸盐一水合物

99%

1229194-11-9

11.

Elagolix

恶拉戈利

99%

834153-87-6

12.

Ivabradine hydrochloride

盐酸依伐布雷定

99%

148849-67-6

13.

Indacaterol maleate

茚达特罗马来酸盐

99%

753498-25-8

14.

Lesinurad

雷西那德

99%

878672-00-5

15.

Liraglutide

利拉鲁肽

99.5%

204656-20-2

16.

Landiolol hydrochloride

盐酸兰地洛尔

99%

144481-98-1

17.

Methotrexate

甲氨蝶呤

USP

59-05-2

18.

Olopatadine hydrochloride

盐酸奥洛他定

USP/99%

140462-76-6

19.

Obeticholic Acid

奥贝胆酸

99%

459789-99-2

20.

Paliperidone palmitate

帕潘立酮棕榈酸酯

99%

199739-10-1

21.

Ropinirole hydrochloride

盐酸罗匹尼罗

99%

91374-20-8

22.

Silodosin

西洛多辛

99%

160970-54-7

23.

Tofacitinib citrate

枸橼酸托法替尼

99%

540737-29-9

24.

Tedizolid phosphate

特地唑胺

99%

856867-55-5

25.

Voglibose

伏格列波糖

99%/JP15

83480-29-9

26.

Nintedanib

尼达尼布

99%

656247-17-5

27.

Lenvatinib mesylate

乐伐替尼甲磺酸盐

99%

857890-39-2

28.

Ponatinib(AP24534)

帕纳替尼

99%

943319-70-8

29.

Lusutrombopag

芦曲泊帕

99%

1110766-97-6

30.

Idelalisib

艾德拉尼

99%

870281-82-6

31.

Crisaborole

克立硼罗

99%

906673-24-3

32.

Niraparib Tosylate Monohydrate

苯甲酸尼拉帕利

99%

1038915-64-8

Intermediates中间体

Intermediates 中间体

No.

Product Name

 

CAS No.

1.

Bepotastine Int. 贝托斯汀中间体

 

2-[(4-Chlorophenyl) (4-piperidinyloxy)methyl]-pyridine

98%

122368-54-1

 

2-[(4-Chlorophenyl)(Piperidin-4-Yloxy) Methyl]-Pyridine,4-Nitrobenzoate(Salt) (1:1)

98%

161558-45-8

 

2-[(S)-(4-chlorophenyl)(4-piperidinyloxy)methyl]pyridine,N-acetyl-L-Phenylalanine(1:1)

99%

210095-66-2

 

2-[(S)-(4-chlorophenyl) (4-piperidinyloxy)methyl]-pyridine

98%

210095-58-2

 

(S)-4-[1-(4-Chlorophenyl)-1-(2-pyridyl) methoxy] piperidine

98%

201594-84-5

2.

Elagolix int.  恶拉戈利中间体

 

Elagolix sodium

99%

832720-36-2

 

5-(2-Fluoro-3-methoxyphenyl)-1-[[2-fluoro-6-(trifluoromethyl)phenyl]methyl]-6-methyl-2,4(1H,3H)-pyrimidinedione

98%

1150560-59-0

 

1-(2-fluoro-6-(trifluoromethyl)benzyl)-5-iodo-6-methylpyrimidine-2,4(1H,3H)-dione

98%

1150560-54-5

 

1-[2-Fluoro-6-(trifluoromethyl)benzyl]-6-methylpyrimidine-2,4(1H,3H)-dione

98%

830346-47-9

 

2,4-Dimethoxy-6-Methyl-Pyrimidine

98%

7781-23-9

 

2-Fluoro-6-(trifluoromethyl)benzyl bromide

98%

239087-08-2

3.

Indacaterol int. 茚达特罗中间体

 

5,6-Diethyl-2,3-dihydro-1H-inden-2-amino Hydrochloride

99%

312753-53-0

 

5-(2R)-2-Oxiranyl-8-benzyloxy-2(1H)-quinolinone

97%

173140-90-4

 

8-Benzyloxy-5-((R)-2-bromo-1-hydroxyethyl)-1H-quinolin-2-one

97%

530084-79-8

 

8-benzyloxy-5-(2-bromoacetyl)-2-(1H)-quinolinone)

98%

100331-89-3

 

2(1H)-Quinolinone,5-[(1R)-2-[(
5,6-diethyl-2,3-dihydro-1H-inden-2-yl)amino]-1-hydroxyethyl]-8-(phenylmethoxy)

98%

435273-75-9

4.

Silodoxin int. 西洛多辛中间体

 

5-[(2R)-2-Aminopropyl]-1-[3-(benzoyloxy)propyl]-2,3-dihydro-1H-indole-7-carbonitrile (2R,3R)-2, 3-dihydroxybutanedioate

98%

239463-85-5

 

2-[2-(2,2,2-Trifluoroethoxy)phenoxy]ethyl methanesulfonate

98%

160969-03-9

5.

Niraparib Tosylate Monohydrate int.苯甲酸尼拉帕利中间体

 

Niraparib HCl

99%

1038915-73-9

 

(S)-tert-butyl 3-(4-aMinophenyl)piperidine-1-carboxylate

99%

1171197-20-8

 

lithium(S)-2-(4-(1-(tert-butoxycarbonyl)piperidin-3-yl)phenyl)-2H-indazole-7-carboxylate

99%

N/A

 

3-Formyl-2-nitrobenzoic acid methyl ester

99%

138229-59-1

6.

Edoxaban  int. 依度沙班中间体

 

tert-Butyl [(1R,2S,5S)-2-amino-5-[(dimethylamino)carbonyl]cyclohexyl]carbamate oxalate

98%

1210348-34-7

 

Tert-Butyl (1R,2S,5S)-2-Amino-5-(Dimethyl Carbamoyl) cyclohexyl-carbamate Oxalate Hydrate

98%

1353893-22-7

 

(1S,3R,4R)-3-(Boc-aMino)-4-hydroxy-cyclohexanecarboxylic acid ethyl ester

98%

365997-33-7

 

5-Methyl-4,5,6,7-tetrahydrothiazolo[5,4-c]pyridine-2-carboxylic acid hydrochloride

98%

720720-96-7

 

2-[(5-Chloropyridin-2-yl)amino]-2-oxoacetic acid ethyl ester monohydrochloride

98%

1243308-37-3

 

N-(5-Chloropyridin-2-yl)oxalamic acid ethyl ester

98%

349125-08-2

7.

Dolutegravir  intermediate:(R)-3-AMINO-1-BUTANOL R-3-氨基丁醇

99%

61477-40-5

8.

Voglibose int. 伏格列波糖中间体

 

2,3,4,6-Tetra-O-benzyl-alpha-D-glucose

98%

6564-72-3

 

Tetrabenzyl-voglibose

98%

115250-39-0

 

(2R,3S,4S,5S)-5-羟基-2,3,4-三(苄氧基)-5-[(苄氧基)甲基]-环己酮

98%

115250-38-9

 

2,3,4,6-Tetra-O-benzyl-D-glucopyranose

98%

4132-28-9

9.

Ivabradine int. 伊伐布雷定中间体

 

3,4-dimethoxy-N-methyl-bicyclo[4.2.0]octa-1,3,5-triene-7-methanamine hydrochloride

99%

866783-13-3

 

3-(3-chloropropyl)-1,3-dihydro-7,8-dimethoxy-2H-3-Benzazepin-2-one

98%

85175-59-3

 

4,5-dimethoxy-1-cyanobenzocyclobutane

98%

35202-54-1

 

7,8-dimethoxy -1,3-dihydro-2H-3-Benzazepin-2-one/2H-3-Benzazepin-2-one, 1,3-dihydro-7,8-dimethoxy

98%

73942-87-7

10.

Lesinurad int.雷西那德中间体

 

lesinurad sodium

99%

1151516-14-1

 

Methyl 2-[[4-(4-cyclopropylnaphthalen-1-yl)-4H-1,2,4-triazol-3-yl]thio]acetate

98%

1533519-85-5

 

3-Amino-4-(4-cyclopropylnaphthalen-1-yl)-4H-1,2,4-triazole-5-thiol

98%

878671-96-6

 

4-(4-cyclopropylnaphthalen-1-yl)-1H-1,2,4-triazole-5(4H)-thione

98%

1533519-84-4

 

1-Cyclopropyl-4-isothiocyanatonaphthalene

98%

878671-95-5

11.

Tedizolid int.  特地唑胺中间体

 

Tedizolid  

99%

856866-72-3

 

N-[3-Fluoro-4-[6-(2-methyl-2H-tetrazol-5-yl)-3-pyridinyl]phenyl]carbamic acid phenylmethyl ester

 

1220910-89-3

 

5-Bromo-2-(2-methyl-2H-tetrazol-5-yl)pyridine

 

380380-64-3

 

(5R)-3-(4-Bromo-3-fluorophenyl)-5-hydroxymethyloxazolidin-2-one

 

444335-16-4

 

2-(2-Methyl-2H-tetrazol-5-yl)pyridine-5-boronic acid pinacol ester

 

1056039-83-8

12.

Lusutrombopag  int. 芦曲泊帕中间体

 

3,5-Dichloro-4-[(1E)-3-ethoxy-2-methyl-3-oxo-1-propen-1-yl]benzoic acid

99%

1110767-89-9

 

(S)-4-(3-(1-(hexyloxy)ethyl)-2-methoxyphenyl)thiazol-2-amine

99%

1110767-98-0

13.

Idelalisib int.艾德拉尼中间体

 

5-fluoro-3-phenyl-2-((1S)-1-((9-(tetrahydro-2H-pyran-2-yl)-9H-purin-6-yl)amino)propyl)quinazolin-4(3H)-one

98%

1453810-71-3

 

(S)-2-(1-aMinopropyl)-5-fluoro-3-phenylquinazolin-4(3H)-one

98%

870281-86-0

 

(S)-tert-butyl(1-(5-fluoro-4-oxo-3-phenyl-3,4-dihydroquinazolin-2-yl)propyl)carbaMate

98%

870281-85-9

14.

Crisaborole int.克立硼罗中间体

 

4-[4-Bromo-3-[[(tetrahydro-2H-pyran-2-yl)oxy]methyl]phenoxy]benzonitrile

98%

943311-78-2

 

4-[4-Bromo-3-[(methoxymethoxy)methyl]phenoxy]benzonitrile

98%

947162-14-3

 

4-[4-Bromo-3-(hydroxymethyl)phenoxy]benzonitrile

98%

906673-45-8

 

4-(4-Bromo-3-formylphenoxy)benzonitrile

98%

906673-54-9

 

4-[4-Bromo-3-(1,3-dioxolan-2-yl)phenoxy]benzonitrile

98%

1217366-74-9

15.

Acotiamide int. 阿考替胺中间体

 

2-Hydroxy-4,5-Dimethoxy Benzoic Acid

98%

5722-93-0

 

Benzoic acid,2-hydroxy-4,5-dimethoxy-,phenyl ester

98%

877997-98-3

 

2-[(2-Hydroxy-4,5-dimethoxybenzoyl)amino]-1,3-thiazole-4-carboxylic acid methyl ester

98%

877997-99-4

16.

Obeticholic Acid int. 奥贝胆酸中间体

 

3α-Hydroxy-7-ketocholanic acid

96%

4651-67-6

 

7-ketolithocholic Methyl ester

96%

10538-59-7

 

(3alpha,5beta,6E)-6-Ethylidene-3-hydroxy-7-oxocholan-24-oic acid

98%

1516887-33-4

17.

Alvimopan int. 爱维莫潘中间体

 

(3R,4R)-3-(3,4-dimethyl-4-piperidiny) phenol

98%

119193-19-0

 

(alphaS,3R,4R)-4-(3-Hydroxyphenyl)-3,4-dimethyl-alpha-(phenylmethyl)-1-piperidinepropanoic acid methyl ester 

98%

170098-29-0

 

(R)-2-Benzyl-3-[(3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethylpiperidin-1-yl]propanoic acid

98%

156130-41-5

 

(S)-2-(((3R,4R)-4-(3-Hydroxyphenyl)-3,4-dimethylpiperidin-1-yl)methyl)-3-phenylpropanoic acid methyl ester hydrochloride

98%

170098-28-9

18.

Ropinirole int. 罗匹尼罗中间体

 

4-(2-Hydroxyethyl)oxyindole

99%

139122-19-3

 

4-[2-[[(4-Methylphenyl)sulfonyl]oxy]ethyl]-2-oxoindole

99%

139122-20-6

19.

Methotrexate int.甲氨蝶呤中间体

 

Methotrexate disodium 

98%

7413-34-5

 

2,4,5,6-Tetraaminopyrimidine sulfate

98%

5392-28-9

 

2,4-diamino-6-(bromomethyl)pteridine

98%

52853-40-4

 

N-[4-(Methylamino)benzoyl]-(L)-Glutamic Acid Diethyl Ester

90%

13726-52-8

 

(2,4-DIAMINOPTERIDIN-6-YL)METHANOL

96%

945-24-4

 

2,4-diamino-6-(hydroxymethyl)-pteridine hydrochloride

95%

73978-41-3

20.

landiolol int. 兰地洛尔中间体

 

4-Hydroxybenzenepropanoic acid [(4S)-2,2-dimethyl-1,3
-dioxolan-4-yl]methyl este

99%

144256-11-1

 

(2S)-(+)Glycidyl-3-nitrobenzene sulfonate

99%

115314-14-2

 

N-(2-aminoethyl)-4-morpholinecarboxamide oxalate

99%

154467-16-0

21.

Tetraisopropyl methylenediphosphonate 亚甲基二磷酸四异丙酯

98%

1660-95-3

22.

Asenapine int. 阿森那平中间体

 

Trans-(+/-)-11-Chloro-2,3,3a,12b-tetrahydro-2-methyl-1H-dibenz[2,3:6,7]oxepino[4,5-c]pyrrole-1-one  

98%

129385-59-7

 

11-chloro-2,3-dihydro-2-methyl-1H-dibenz[2,3;6,7]oxepino[4,5-c]pyrrol-1-one

98%

1012884-46-6

23.

Dabigatran int. 达比加群中间体

 

Dabigatran etexilate 

99%

211915-06-9

 

3-[(3-Amino-4-methylaminobenzoyl)pyridin-2-ylamino]propionic acid ethyl ester 

98%

212322-56-0

 

N-(4-Cyanophenyl)glycine 

98%

42288-26-6

 

3-[[[2-[[(4-Cyanophenyl)amino]methyl]-1-methyl-1H-benzimidazol-5-yl]carbonyl]pyridin-2-ylamino]propionic acid ethyl ester

98%

211915-84-3

24.

Nabilone int. 那密浓中间体

 

2-(4-Methoxy-1,4-cyclohexadienyl)-2-propanol

97%

61597-37-3

 

5-(1,1-Dimethylheptyl)resorcinol

97%

56469-10-4


杂质列表

沃诺拉赞杂质

西格列汀杂质

索非布韦杂质

基因毒性杂质

多索茶碱杂质

咪达唑仑杂质

阿戈美拉汀杂质

甲磺酸乙酯

特地唑胺杂质

LCZ696杂质

替诺福韦拉酚氨酯(替诺福韦艾拉酚胺)杂质

甲磺酸甲酯

帕立骨化醇杂质

托法替尼杂质

西那卡塞杂质

对甲苯磺酸正丁酯

美托洛尔杂质

奥卡西平杂质

普瑞巴林杂质

对甲苯磺酸异丙酯

恩替卡韦杂质

氟吡汀杂质

伊马替尼杂质

对甲苯磺酸乙酯

度洛西汀杂质

帕利哌酮杂质

依度沙班杂质

对甲苯磺酸甲酯

帕瑞昔布钠杂质

尼达尼布杂质

阿加曲班杂质

甲磺酸异丙酯

头孢唑林钠杂质

瑞舒伐他汀钙杂质

阿普斯特杂质

对甲苯磺酸正丁酯

长春西汀杂质

伊伐布雷定杂质

阿考替胺杂质

托法替尼

厄洛替尼杂质

布洛芬杂质

奥氮平杂质

利奥西呱

非布索坦杂质

氨溴索杂质

依折麦布杂质

帕瑞昔布钠

双丙戊酸钠杂质

阿齐沙坦酯杂质

利伐沙班杂质

托法替尼  

替格瑞洛杂质

帕布昔利布杂质

奥美拉唑杂质

西那卡塞

埃索美拉唑杂质

兰索拉唑杂质

雷贝拉唑杂质

莫西沙星

泮托拉唑杂质

丁酸氯维地平杂质

氨氯地平杂质

埃索(奥美)拉唑

非洛地平杂质

硝苯地平杂质

阿哌沙班杂质

 

氟康唑杂质

福司氟康唑杂质

莫西沙星杂质

 

左氧氟沙星杂质

非马沙坦杂质

缬沙坦杂质

 

阿齐沙坦杂质

奥美沙坦酯杂质

氯沙坦钾杂质

 

奥拉西坦杂质

左乙拉西坦杂质

达比加群酯杂质

 

依达拉奉杂质

纳美芬杂质

考尼伐坦杂质

 

罗氟司特杂质

雷美替胺杂质

阿法替尼杂质

 

替诺福韦酯杂质

曲格列汀杂质

阿格列汀杂质

 

普萘洛尔杂质

沃拉帕沙杂质

门冬氨酸鸟氨酸杂质

 

普拉克索杂质

卡培他滨杂质

利格列汀杂质

 

硝呋太尔杂质

多塞平杂质

氯吡格雷杂质

 

吉非替尼杂质

依托咪酯杂质

阿托伐他汀钙杂质


     
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